Data di Pubblicazione:
2023
Abstract:
A targeted bibliographic search exposed the deficiencies within existing PROTAC preclinical pipelines, including missing, poor-quality data and technical limitations in the experimental assays. Several recommendations are proposed to improve the efficiency of preclinical platforms for PROTACs.
Tipologia CRIS:
03A-Articolo su Rivista
Keywords:
Permeability; Physicochemical descriptors; Preclinical pipeline; PROTAC; Solubility
Elenco autori:
Apprato, Giulia; Ermondi, Giuseppe; Caron, Giulia
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